Futibatinib

First covalent (irreversible) pan-FGFR inhibitor; overcomes FGFR resistance mutations. Only covalent FGFR inhibitor — overcomes FGFR resistance point mutations

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Description

Scientific Overview: First covalent (irreversible) pan-FGFR inhibitor; overcomes FGFR resistance mutations. Only covalent FGFR inhibitor — overcomes FGFR resistance point mutations

Mechanism of Action: FGFR1/2/3/4 Covalent Inhibitor

Purity: ≥99%  |  Molecular Formula: C24H26F2N4O4S

For Research Use Only. Not intended for diagnostic, therapeutic, or clinical applications.

Additional information

Effect

FGFR1/2/3/4 Covalent Inhibitor

Purity

≥99%

Molecular Formula

C24H26F2N4O4S

CAS Number

1448997-69-0